SCHEMBL17545211

SCHEMBL17545211

CC(=O)N1CCc2cc(Cl)c(S(=O)(=O)Nc3ccc(C)cn3)cc21

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 5/20 0.47
NOTUM Q6P988 3/20 0.46
KMT2A Q03164 2/20 0.46
PKM P14618 2/20 0.46
LMNA P02545 1/20 0.46
MEN1 O00255 1/20 0.46
NR3C1 P04150 1/20 0.44
CYP11B2 P19099 1/20 0.44
ACLY P53396 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19219760 0.91 KMT2A (0.41) TRIM24KMT2APKMLMNAMEN1
SCHEMBL17545074 0.85 KMT2A (0.52) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL17545073 0.83 CYP11B2 (0.52) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL17545288 0.80 LMNA (0.50) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL15882573 0.78 NOTUM (0.51) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL29707960 0.78 NOTUM (0.51) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL17545149 0.77 USP2 (0.53) TRIM24KMT2APKMLMNACYP11B2
SCHEMBL19219758 0.76 KDM4E (0.46) TRIM24KMT2APKMLMNAMEN1
SCHEMBL23613816 0.75 KMT2A (0.48) TRIM24NOTUMKMT2APKMLMNA
SCHEMBL15882287 0.74 NOTUM (0.55) TRIM24NOTUMKMT2APKMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180312-B1 INDOLINE SULFONAMIDE INHIBITORS OF DAPE AND NDM-1 AND USE OF THE SAME UNIV LOYOLA CHICAGO (US) 2019-10-16 EP disclosed
US-10385040-B2 Indoline sulfonamide inhibitors of DapE and NDM-1 and use of the same LOYOLA UNIVERSITY OF CHICAGO (US) 2019-08-20 US disclosed
US-20170226090-A1 INDOLINE SULFONAMIDE INHIBITORS OF DAPE AND NDM-1 AND USE OF THE SAME BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2017-08-10 US disclosed
WO-2016025637-A1 INDOLINE SULFONAMIDE INHIBITORS OF DAPE AND NDM-1 AND USE OF THE SAME LOYOLA UNIVERSITY OF CHICAGO (US) 2016-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10385040-B2 Indoline sulfonamide inhibitors of DapE and NDM-1 and use of the same INMT, MGAM, NNMT TRIM24 1559/4885NOTUM 581/4885KMT2A 1720/4885
US-20170226090-A1 INDOLINE SULFONAMIDE INHIBITORS OF DAPE AND NDM-1 AND USE OF THE SAME INMT, MGAM, NNMT TRIM24 1559/4885NOTUM 581/4885KMT2A 1720/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.