SCHEMBL175765

SCHEMBL175765

COC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)c1ccc(C#CC#Cc2ccc(N)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.39
TAS1R1 Q7RTX1 4/20 0.39
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
LNPEP Q9UIQ6 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15227743 0.85 RAB9A (0.44) TAS1R3TAS1R1GAARAB9AL3MBTL1
SCHEMBL403947 0.85 PTPN11 (0.38) TAS1R3TAS1R1GAARAB9ALNPEP
SCHEMBL1105518 0.85 PTPN11 (0.38) TAS1R3TAS1R1GAARAB9ALNPEP
SCHEMBL9087370 0.85 EPHX2 (0.43) GAARAB9AADRB2ADRB1ADRB3
SCHEMBL9087368 0.85 EPHX2 (0.43) GAARAB9AADRB2ADRB1ADRB3
SCHEMBL15227850 0.81
SCHEMBL19684300 0.78 TAS1R3 (0.40) TAS1R3TAS1R1GAARAB9ALNPEP
SCHEMBL13245476 0.78 L3MBTL1 (0.50) TAS1R3TAS1R1GAARAB9ALNPEP
SCHEMBL28940166 0.78 TAS1R3 (0.45) TAS1R3TAS1R1GAARAB9ALNPEP
SCHEMBL20299887 0.78 TAS1R3 (0.45) TAS1R3TAS1R1GAARAB9ALNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed