SCHEMBL1759104

SCHEMBL1759104

O=C(O)c1cc2ccccn2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.49
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
DAO P14920 1/20 0.43
TSHR P16473 1/20 0.43
NAPRT Q6XQN6 1/20 0.43
KDM4E B2RXH2 3/20 0.42
NPC1 O15118 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
POLB P06746 3/20 0.42
ALOX15 P16050 1/20 0.41
IMPDH2 P12268 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SSTR4 P31391 1/20 0.38
CES2 O00748 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559325 0.85 CHRNA7 (0.49) CHRNA7PTGS1PTGS2KDM4ENPC1
SCHEMBL12647211 0.83 CHRNA7 (0.48) CHRNA7KDM4ENPC1ALDH1A1MAPT
SCHEMBL1421391 0.83 CHRNA7 (0.48) CHRNA7TSHRKDM4ENPC1ALDH1A1
Hydrochloric Acid SCHEMBL1421587 0.81 CHRNA7 (0.47) CHRNA7TSHRKDM4ENPC1ALDH1A1
SCHEMBL27972521 0.79 KMO (0.49) DAOTSHRNAPRTMAPTSMN1; SMN2
SCHEMBL14669997 0.79 CHRNA7 (0.45) CHRNA7PTGS1PTGS2TSHRKDM4E
SCHEMBL12060479 0.79 CHRNA7 (0.45) CHRNA7TSHRKDM4ENPC1ALDH1A1
SCHEMBL28907062 0.79 GSK3B (0.48) CHRNA7KDM4ENPC1ALDH1A1MAPT
SCHEMBL25514718 0.79 CHRNA7 (0.45) CHRNA7PTGS1PTGS2KDM4ENPC1
SCHEMBL25514623 0.79 CHRNA7 (0.45) CHRNA7PTGS1PTGS2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 126 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120157670-A Indolizine-2-carboxylic acid derivative and preparation method and application thereof 浙江大学 2025-06-17 CN claimed
EP-3710428-B1 MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2026-03-25 EP disclosed
EP-4662208-A1 COMPOUNDS AND COMPOSITIONS FOR SELECTIVE DEGRADATION OF ENGINEERED PROTEINS Celgene Corporation (US) 2025-12-17 EP disclosed
CN-120157670-A Indolizine-2-carboxylic acid derivative and preparation method and application thereof 浙江大学 2025-06-17 CN disclosed
CN-120157670-A Indolizine-2-carboxylic acid derivative and preparation method and application thereof 浙江大学 2025-06-17 CN disclosed
CN-120157670-A Indolizine-2-carboxylic acid derivative and preparation method and application thereof 浙江大学 2025-06-17 CN disclosed
US-20240327381-A1 Compounds and Compositions for Selective Degradation of Engineered Proteins CELGENE CORPORATION (US) 2024-10-03 US disclosed
US-20240307382-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ABBVIE INC. 2024-09-19 US disclosed
WO-2024167999-A1 COMPOUNDS AND COMPOSITIONS FOR SELECTIVE DEGRADATION OF ENGINEERED PROTEINS CELGENE CORPORATION (US) 2024-08-15 WO disclosed
US-20240228504-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2024-07-11 US disclosed
WO-2003048123-A1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-06-12 WO disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed
WO-2000026177-A1 SYNTHESIS OF ETHYL BROMOPYRUVATE GREAT LAKES CHEMICAL CORPORATION (US) 2000-05-11 WO disclosed
EP-0998488-A1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2000-05-10 EP disclosed
EP-0988303-A1 PYRROLO 2,1,5-cd]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 2000-03-29 EP disclosed
WO-1999002549-A1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-01-21 WO disclosed
WO-1998055483-A1 PYRROLO[2,1,5-cd]INDOLIZINE DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES NOVO NORDISK A/S (DK) 1998-12-10 WO disclosed
US-5756501-A USEFUL FOR TREATING ALZHIMER'S DISEASE, DOWN'S SYNDROM AND PARKINSON'S DISEASE INVOLVING HYPOFUNCTION OF ACETYLCHOLINE IN MAMMAL AMERICAN HOME PRODUCTS CORPORATION (US) 1998-05-26 US disclosed
WO-1991010664-A1 PYRIDAZINO[4,5-b]INDOLIZINES AMERICAN HOME PRODUCTS CORPORATION (US) 1991-07-25 WO disclosed
US-4985560-A Pyridazino(4,5-b)indolizines AMERICAN HOME PRODUCTS CORPORATION (US) 1991-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240327381-A1 Compounds and Compositions for Selective Degradation of Engineered Proteins TP53, APC, MDM2 CHRNA7 4861/4885PTGS1 3832/4885PTGS2 3791/4885
US-20240228504-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME SLC10A1, NR1H4, SLC10A2 CHRNA7 4831/4885PTGS1 3990/4885PTGS2 4376/4885
US-20240307382-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ATF4, ATF1, DDIT3 CHRNA7 4444/4885PTGS1 321/4885PTGS2 324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.