Pyrrolidine

Pyrrolidine

SCHEMBL17599458

C1CCNC1.NS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.73

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.73
CA9 Q16790 2/20 0.73
CA2 P00918 2/20 0.73
PNMT P11086 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CDK2 P24941 1/20 0.47
HTR6 P50406 6/20 0.45
F2 P00734 2/20 0.45
PRSS1 P07477 2/20 0.45
PRSS2 P07478 2/20 0.45
PRSS3 P35030 2/20 0.45
LDHA P00338 1/20 0.43
CA12 O43570 1/20 0.43
TSHR P16473 1/20 0.43
ROCK2 O75116 2/20 0.42
CCR2 P41597 2/20 0.42
ROCK1 Q13464 2/20 0.42
CIT O14578 1/20 0.42
DAPK3 O43293 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29529240 0.86 CA2 (1.00) CA1CA9CA2MEN1KMT2A
SCHEMBL28464 0.86 CA2 (1.00) CA1CA9CA2MEN1KMT2A
Benzene SCHEMBL11062753 0.84 CA2 (0.96) CA1CA9CA2MEN1KMT2A
SCHEMBL27901054 0.84 CA2 (0.96) CA1CA9CA2MEN1KMT2A
Hydrochloric Acid SCHEMBL951327 0.84 CA2 (0.96) CA1CA9CA2MEN1KMT2A
Ammonia Solution, Strong SCHEMBL28028391 0.84 CA2 (0.96) CA1CA9CA2MEN1KMT2A
Hydrochloric Acid SCHEMBL8125684 0.82 CA2 (0.92) CA1CA9CA2MEN1KMT2A
Phosphoric Acid SCHEMBL28841729 0.77 CA2 (0.81) CA1CA9CA2MEN1KMT2A
Acetamide SCHEMBL28617889 0.76 CA2 (0.79) CA1CA9CA2CDK2HTR6
Isothiocyanate SCHEMBL28619475 0.76 CA2 (0.79) CA1CA9CA2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110511170-A A kind of synthetic method of chirality nafoxidine -3- carboxylic acid HANGZHOU ALLSINO BIOTECHNOLOGY CO LTD 2019-11-29 CN disclosed
EP-2997966-A1 Naphthyl Sulfonamide Pyrrolidine Derivatives as KEAP-1 Modulators for the Treatment of Diabetes, Obesity, Dyslipidemia and Related Disorders SANOFI (FR) 2016-03-23 EP disclosed
EP-2997966-A1 Naphthyl Sulfonamide Pyrrolidine Derivatives as KEAP-1 Modulators for the Treatment of Diabetes, Obesity, Dyslipidemia and Related Disorders SANOFI (FR) 2016-03-23 EP disclosed