SCHEMBL17609773

SCHEMBL17609773

Cc1ncc(C(F)(F)F)cc1-c1cccc(N)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.39
SCN9A Q15858 1/20 0.39
MPL P40238 1/20 0.37
ASIC3 Q9UHC3 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
NOS3 P29474 4/20 0.36
NOS2 P35228 3/20 0.36
FEN1 P39748 3/20 0.36
ALOX5AP P20292 2/20 0.36
NOS1 P29475 3/20 0.36
BACE1 P56817 1/20 0.36
BRD4 O60885 1/20 0.35
KDM1A O60341 1/20 0.35
HPGD P15428 1/20 0.35
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17610099 0.74 ASIC3 (0.44) ASIC3BACE1KDM1APIK3CD
SCHEMBL26522084 0.74 ASIC3 (0.42) ASIC3NOS3NOS2FEN1ALOX5AP
SCHEMBL26650965 0.72 MET (0.48) METCYP2C19ADORA2AADORA1
SCHEMBL18039077 0.72 ASIC3 (0.47) ASIC3ADORA2AADORA1BACE1KDM1A
SCHEMBL17619753 0.70 ASIC3 (0.45) ASIC3NOS3NOS2ALOX5APKDM1A
SCHEMBL6256565 0.69 CTSS (0.60) ASIC3ADORA2AADORA1BRD4KDM1A
SCHEMBL30797381 0.69 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19NOS3NOS2
SCHEMBL573513 0.69 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19NOS3NOS2
SCHEMBL29464843 0.69 SCN9A (0.40) METSCN9AMPLCYP1A2CYP3A4
SCHEMBL28715902 0.69 SCN9A (0.40) METSCN9AMPLCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3193880-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Hydra Biosciences, Inc. (US) 2017-07-26 EP disclosed
WO-2016044792-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2016-03-24 WO disclosed