SCHEMBL17620844

SCHEMBL17620844

NC(=O)N1CC(c2cccnn2)C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 2/20 0.48
PDE9A O76083 2/20 0.38
P2RX7 Q99572 1/20 0.37
CYP1A2 P05177 1/20 0.33
FAAH O00519 3/20 0.33
SLC6A7 Q99884 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
LTA4H P09960 1/20 0.32
HSD11B1 P28845 1/20 0.32
NAMPT P43490 1/20 0.31
PARP1 P09874 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1740371 0.85 KDM5A (0.46) KDM5APDE9AP2RX7CYP1A2FAAH
SCHEMBL2993386 0.77 GPR119 (0.44) KDM5ANAMPT
SCHEMBL13075972 0.74 KDM5A (0.39) KDM5APDE9ACHRNB4CHRNA3CHRNA7
SCHEMBL17620811 0.72 KDM5A (0.37) KDM5AP2RX7CYP1A2SLC6A7
SCHEMBL1963995 0.72 PRMT5 (0.39) KDM5A
SCHEMBL15529416 0.71 NAMPT (0.60) KDM5ANAMPT
SCHEMBL17675448 0.71 CYP11B2 (0.42) KDM5APDE9A
SCHEMBL29765569 0.70
SCHEMBL16060787 0.70
SCHEMBL3393553 0.70 GOT1 (0.37) KDM5APDE9AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296723-B2 NAMPT inhibitors ABBVIE INC. (US) 2016-03-29 US disclosed