SCHEMBL17624705

SCHEMBL17624705

CCCc1cccc(C(=O)NNC(C)(C)C)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 1/20 0.38
HCRTR1 O43613 4/20 0.37
HCRTR2 O43614 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
HTT P42858 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KAT6A Q92794 1/20 0.35
CTSS P25774 1/20 0.34
HPGD P15428 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HSD17B10 Q99714 1/20 0.34
F2R P25116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28277840 0.90 KAT6A (0.40) CD38SMN1; SMN2HTTKAT6ACTSS
SCHEMBL17625005 0.80 CTSS (0.36) CD38HCRTR1HCRTR2SMN1; SMN2HTT
SCHEMBL8174016 0.79 NPC1 (0.46) CD38SMN1; SMN2HTTCYP1A2CYP3A4
SCHEMBL28642784 0.76 GABRA1 (0.39) HCRTR1HCRTR2HTTCYP1A2CYP3A4
SCHEMBL7045375 0.76 EZH2 (0.49) HCRTR1ALDH1A1
SCHEMBL2362450 0.75 MRGPRX4 (0.47) HTTHPGDCA9HSD17B10KDM4E
SCHEMBL22620361 0.75 PRKCI (0.42) HCRTR1HCRTR2HTTCYP1A2CYP3A4
SCHEMBL8174111 0.74 HPGD (0.53) SMN1; SMN2HTTKAT6AHPGDNPC1
SCHEMBL29778078 0.74 ABCB1 (0.52) SMN1; SMN2NPC1RAB9A
SCHEMBL28276332 0.74 KCNK3 (0.40) SMN1; SMN2HTTCYP1A2CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016044390-A1 BORON-CONTAINING DIACYLHYDRAZINE COMPOUNDS INTREXON CORPORATION (US) 2016-03-24 WO disclosed