SCHEMBL17629944

SCHEMBL17629944

N#Cc1ccc(-c2ncc(I)cc2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.40
RHEB Q15382 1/20 0.39
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
KDM1A O60341 5/20 0.38
GRM5 P41594 1/20 0.38
PTPN11 Q06124 1/20 0.37
RIPK1 Q13546 1/20 0.37
CYP11B2 P19099 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
NSD2 O96028 1/20 0.36
MMP3 P08254 1/20 0.35
MAOB P27338 1/20 0.35
MALT1 Q9UDY8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17630030 0.81 PLAU (0.43) PLAURHEBKDM1AGRM5PTPN11
SCHEMBL17629890 0.78 CYP11B2 (0.41) CYP11B2NSD2
SCHEMBL17630009 0.78 EGLN2 (0.40) KDM1AGRM5CYP11B2NSD2
SCHEMBL17630044 0.77 KDM1A (0.41) KDM1APTPN11CYP11B2NSD2MAOB
SCHEMBL17629945 0.75 VCAM1 (0.47) PLAUTDP1
SCHEMBL9140783 0.75 RHEB (0.42) PLAURHEBGSK3BCYP11B2NSD2
SCHEMBL17630012 0.74 MMP3 (0.41) PLAURHEBCCNB2CDK1CCNB1
SCHEMBL17630026 0.71 KDM1A (0.41) RHEBKDM1ACYP11B2NSD2MMP3
SCHEMBL10061101 0.71 SLC22A12 (0.48) RHEBCYP11B2
SCHEMBL17630049 0.71 ADH5 (0.65) CYP11B2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016046782-A1 IMIDAZOLE BIARYL COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-03-31 WO disclosed