SCHEMBL17632277

SCHEMBL17632277

NC(=O)c1ccc(Cl)c(-c2noc([CH]COCc3ccccc3)n2)c1Cl

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
CNR1 P21554 1/20 0.34
WEE1 P30291 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PARP10 Q53GL7 1/20 0.32
ATM Q13315 2/20 0.32
KMT2A Q03164 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
GSTP1 P09211 2/20 0.32
FFAR1 O14842 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK14 Q16539 1/20 0.31
ADRA1D P25100 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17632072 0.82 NPC1 (0.48) NPC1RAB9APARP10ATMALDH1A1
SCHEMBL4248899 0.81 SENP7 (0.37) NPC1RAB9AKMT2ASENP7ALDH1A1
SCHEMBL17513876 0.79 GRM5 (0.39) NPC1RAB9APARP10SENP7PARP1
SCHEMBL17514018 0.74 KMT2A (0.35) NPC1RAB9AKDM4EATMKMT2A
SCHEMBL17513938 0.73 CA12 (0.39) NPC1RAB9AATMFFAR1ALDH1A1
SCHEMBL4988520 0.69 SIRT2 (0.43) NPC1KDM4EPARP10KMT2AALDH1A1
SCHEMBL17513978 0.68 ATM (0.41) NPC1RAB9AATMSENP7ALDH1A1
SCHEMBL8885349 0.64 KMT2A (0.53) WEE1KDM4EATMKMT2AALDH1A1
SCHEMBL4986019 0.63 CYP3A4 (0.43) NPC1RAB9AKDM4EKMT2AALDH1A1
SCHEMBL17514014 0.63 ATM (0.53) NPC1RAB9AATMKMT2ASENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197482-A1 METHODS OF TREATING TRAUMATIC BRAIN INJURY Oxeia Biopharmaceuticals Inc. (US) 2017-08-02 EP disclosed
WO-2016048488-A1 METHODS OF TREATING TRAUMATIC BRAIN INJURY OXEIA BIOPHARMACEUTICALS, INC. (US) 2016-03-31 WO disclosed