SCHEMBL1763732

SCHEMBL1763732

N#Cc1ccccc1C(=O)N1CC=C(c2ccc(C(=O)NC(=N)NC(=O)OCc3ccccc3)cc2C(F)(F)F)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
SLC9A1 P19634 1/20 0.39
CYP2C19 P33261 1/20 0.39
PTGDR2 Q9Y5Y4 6/20 0.36
BTK Q06187 4/20 0.35
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
HSD11B1 P28845 1/20 0.33
SCD O00767 1/20 0.33
SMO Q99835 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1764093 0.84 CYP2C9 (0.48) CYP2D6CYP2C9SLC9A1CYP2C19MMP2
SCHEMBL1763602 0.84 P2RX7 (0.39) SLC9A1PTGDR2BTKMMP2MMP3
SCHEMBL1763534 0.83 BTK (0.41) PTGDR2BTKMMP2MMP3MAPT
SCHEMBL12593569 0.74 NAMPT (0.40) CYP2D6CYP2C9SLC9A1CYP2C19HSD11B1
SCHEMBL1763801 0.72 SLC9A1 (0.55) CYP2D6CYP2C9SLC9A1CYP2C19
SCHEMBL1763651 0.72 SLC9A1 (0.46) CYP2D6CYP2C9SLC9A1CYP2C19HSD11B1
SCHEMBL1763592 0.70 SLC9A1 (0.49) SLC9A1MMP2MMP3MAPT
SCHEMBL1763934 0.70 SLC9A1 (0.54) CYP2D6CYP2C9SLC9A1CYP2C19
SCHEMBL1763563 0.69 SLC9A1 (0.51) CYP2D6CYP2C9SLC9A1CYP2C19KMT2A
SCHEMBL1840448 0.69 PTGDR2 (0.38) PTGDR2BTKMMP2MMP3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110118262-A1 Pyrrolidinyl and Piperidinyl Compounds Useful as NHE-1 Inhibitiors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118262-A1 Pyrrolidinyl and Piperidinyl Compounds Useful as NHE-1 Inhibitiors NHERF1, SLC9A1, SLC9A5 CYP2D6 2007/4885CYP2C9 1660/4885SLC9A1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.