SCHEMBL17644142

SCHEMBL17644142

[CH]c1cccc(N2CCN(c3ccncc3)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.52
ADRB2 P07550 1/20 0.47
NCF1 P14598 1/20 0.47
PLD1 Q13393 1/20 0.47
KHK P50053 4/20 0.46
AOC3 Q16853 2/20 0.45
MAPT P10636 4/20 0.43
PLOD2 O00469 2/20 0.43
PLOD3 O60568 2/20 0.43
PLOD1 Q02809 2/20 0.43
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
LMNA P02545 1/20 0.42
EED O75530 1/20 0.41
DHFR P00374 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7589729 0.80 ADRA2C (0.62) CHKAADRB2NCF1PLD1KHK
SCHEMBL7398706 0.79 DRD2 (0.55) CHKAADRB2NCF1PLD1KHK
SCHEMBL18590696 0.78 CHKA (0.67) CHKAADRB2NCF1PLD1KHK
SCHEMBL28112415 0.78 CHKA (0.80) CHKAADRB2NCF1PLD1MAPT
SCHEMBL7398283 0.76 MAPT (0.69) KHKMAPTKDM4EGAADHFR
SCHEMBL12525660 0.75 AOC3 (0.57) CHKAADRB2NCF1PLD1KHK
SCHEMBL8634506 0.72 CHKA (0.64) CHKAADRB2NCF1PLD1MAPT
SCHEMBL49273 0.69 CHKA (1.00) CHKAADRB2NCF1PLD1MAPT
SCHEMBL19468905 0.69 CHKA (0.90) CHKAADRB2NCF1PLD1MAPT
SCHEMBL23035473 0.69 CHKA (0.64) CHKAADRB2NCF1PLD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002278-A1 GUANIDINE COMPOUND Astellas Pharma Inc. (JP) 2016-04-06 EP disclosed