SCHEMBL17656334

SCHEMBL17656334

O=CC1(c2ccc3c(c2)CCO3)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.44
DYRK1A Q13627 6/20 0.43
DYRK1B Q9Y463 5/20 0.43
DYRK2 Q92630 3/20 0.43
PRKCI P41743 1/20 0.41
SLC6A2 P23975 5/20 0.40
SLC6A4 P31645 5/20 0.40
CLK1 P49759 3/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
CLK2 P49760 1/20 0.40
CLK3 P49761 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19594729 0.87 CHRM2 (0.42) ERN1DYRK1ADYRK1BDYRK2PRKCI
SCHEMBL8895190 0.81 LMNA (0.47) DYRK1ADYRK1BDYRK2SLC6A2SLC6A4
SCHEMBL9587145 0.75 ALDH1A1 (0.50) SLC6A4HDAC3HDAC1HDAC2HDAC6
SCHEMBL13458449 0.75 PRKCI (0.45) ERN1DYRK1ADYRK1BDYRK2PRKCI
SCHEMBL1465591 0.73 SLC6A2 (0.44) ERN1PRKCISLC6A2SLC6A4HDAC3
SCHEMBL13365167 0.72 SLC6A2 (0.46) ERN1PRKCISLC6A2SLC6A4HDAC3
SCHEMBL21907080 0.71 PRKCI (0.45) ERN1DYRK1ADYRK1BDYRK2PRKCI
SCHEMBL12742727 0.71 DYRK1A (0.44) ERN1DYRK1ADYRK1BDYRK2PRKCI
SCHEMBL339129 0.70 DYRK1A (0.61) ERN1DYRK1ADYRK1BDYRK2PRKCI
SCHEMBL12825139 0.69 PIK3CA (0.42) PIK3CANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2674428-B1 Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2016-04-06 EP disclosed