SCHEMBL17656383

SCHEMBL17656383

N#CC1(c2ccc3c(c2)CCC(F)(F)CC3)CC1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.40
KMT2A Q03164 1/20 0.35
WDR5 P61964 2/20 0.35
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1466762 0.86 OPRM1 (0.44) OPRM1KMT2AWDR5PDE4APDE4B
SCHEMBL13362358 0.73 OPRM1 (0.38) OPRM1KMT2AWDR5CYP1A2
SCHEMBL21874208 0.71 WDR5 (0.41) OPRM1WDR5
SCHEMBL24214281 0.70 OPRM1 (0.40) OPRM1WDR5CYP1A2
SCHEMBL10209132 0.69 OPRM1 (0.51) OPRM1KMT2A
SCHEMBL2200912 0.69 SLC6A4 (0.43) OPRM1KMT2AWDR5
SCHEMBL14711714 0.69 OPRM1 (0.44) OPRM1KMT2A
SCHEMBL4515335 0.68 OPRM1 (0.41) OPRM1KMT2ACYP1A2
SCHEMBL16526958 0.67 ADRA2A (0.45)
SCHEMBL2937652 0.67 KDM1A (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2674428-B1 Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2016-04-06 EP disclosed