SCHEMBL17656572

SCHEMBL17656572

O=C(O)c1ccccc1C1=NC=CCN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
RAB9A P51151 3/20 0.40
ALDH1A1 P00352 7/20 0.39
ALOX15 P16050 2/20 0.39
MYC P01106 1/20 0.39
POLB P06746 1/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX12 P18054 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
TSHR P16473 2/20 0.37
USP2 O75604 1/20 0.37
HNF4A P41235 1/20 0.37
GAA P10253 1/20 0.36
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
FOLH1 Q04609 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11081413 0.73 FABP4 (0.47) KDM4EALDH1A1POLBCYP3A4CYP2C9
SCHEMBL29726703 0.72 ALDH1A1 (0.52) KDM4ERAB9AALDH1A1ALOX15MYC
SCHEMBL7799064 0.72 ALDH1A1 (0.52) KDM4ERAB9AALDH1A1ALOX15MYC
SCHEMBL1526540 0.71 NISCH (0.60)
SCHEMBL8376104 0.70 KDM4E (0.41) KDM4ERAB9AALDH1A1ALOX15MYC
SCHEMBL7488646 0.69 NISCH (0.56) KDM4ERAB9AALDH1A1ALOX15MYC
SCHEMBL36145 0.69 ALDH1A1 (0.72) KDM4EALDH1A1ALOX15MYCPOLB
SCHEMBL30028907 0.69 ALDH1A1 (0.72) KDM4EALDH1A1ALOX15MYCPOLB
SCHEMBL7486584 0.68 NISCH (0.50) KDM4ERAB9AALDH1A1CYP3A4CYP2C9
SCHEMBL2029224 0.67 ALDH1A1 (0.41) KDM4ERAB9AALDH1A1ALOX15MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632253-B1 PROCESS FOR THE PREPARATION OF AN OREXIN RECEPTOR ANTAGONIST MERCK SHARP & DOHME (US) 2016-04-06 EP disclosed