SCHEMBL17664014

SCHEMBL17664014

Fc1ccc(Cc2ncc(Cl)cc2Cl)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
FYN P06241 1/20 0.35
MAPK14 Q16539 1/20 0.35
LMNA P02545 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
APEX1 P27695 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MPO P05164 1/20 0.34
KDM5A P29375 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
CNR1 P21554 2/20 0.33
EGFR P00533 2/20 0.33
CNR2 P34972 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17663880 0.82 HSP90AB1 (0.40) MEN1KMT2ALMNACYP2C9TSHR
SCHEMBL17664085 0.82 PARP1 (0.37) PARP1LMNACYP2C9TSHRAPEX1
SCHEMBL17664049 0.78 PARP1 (0.35) PARP1EGFR
SCHEMBL17663941 0.76 MEN1 (0.39) PARP1MEN1KMT2ACYP17A1CYP11B1
SCHEMBL17664078 0.75 MEN1 (0.39) PARP1MEN1KMT2ALMNAALDH1A1
SCHEMBL17664100 0.75 FYN (0.41) CYP17A1CYP11B1CYP11B2FYNMAPK14
SCHEMBL17664012 0.74 SMN1; SMN2 (0.50) MEN1KMT2ALMNACYP2C9TSHR
SCHEMBL23716083 0.72 TDP1 (0.35) PARP1MEN1KMT2ACYP17A1CYP11B1
SCHEMBL23715848 0.72 RAB9A (0.38) MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL3299911 0.71 CYP17A1 (0.52) CYP17A1CYP11B1CYP11B2MPOKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed
WO-2016053855-A1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-04-07 WO disclosed