SCHEMBL17664100

SCHEMBL17664100

Fc1ccc(Cc2ccc(Cl)cn2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.41
CYP17A1 P05093 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
HSP90AB1 P08238 1/20 0.37
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
MPO P05164 1/20 0.35
MBOAT4 Q96T53 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
KDM5A P29375 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
CNR1 P21554 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.34
METAP2 P50579 1/20 0.34
DAO P14920 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664001 0.90 GPR52 (0.35) FYNHSP90AB1MBOAT4KDM4EDAO
SCHEMBL17664358 0.88 HDAC3 (0.41) HSP90AB1DAO
SCHEMBL23716215 0.87 MBOAT4 (0.37) FYNHSP90AB1MBOAT4KDM4EDAO
SCHEMBL23716265 0.85 RXRA (0.39) HSP90AB1MPOMBOAT4DAO
SCHEMBL17663971 0.81 HSP90AB1 (0.47) HSP90AB1MBOAT4ALDH1A1KDM4E
SCHEMBL17663857 0.81 IDO1 (0.42) HSP90AB1ALDH1A1HTT
SCHEMBL23716203 0.80 MBOAT4 (0.39) HSP90AB1MBOAT4S1PR1S1PR3ALDH1A1
SCHEMBL17664376 0.77 ALDH1A1 (0.43) MBOAT4ALDH1A1HTTKDM4EMAPK14
SCHEMBL23716095 0.76 GPR52 (0.34) FYNKDM5AKDM5B
SCHEMBL17663975 0.75 RAB9A (0.48) HSP90AB1MBOAT4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed
WO-2016053855-A1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-04-07 WO disclosed