SCHEMBL17664012

SCHEMBL17664012

COc1ccc(Cc2ncc(Cl)cc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.50
LMNA P02545 2/20 0.50
ALDH1A1 P00352 1/20 0.50
TSHR P16473 2/20 0.47
CYP2C9 P11712 1/20 0.47
APEX1 P27695 1/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 2/20 0.47
ALOX5 P09917 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
PDE10A Q9Y233 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
LTA4H P09960 1/20 0.43
KDR P35968 3/20 0.43
MAPK1 P28482 2/20 0.42
MDM4 O15151 1/20 0.41
TP53 P04637 1/20 0.41
MDM2 Q00987 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL23716277 0.85 ALDH1A1 (0.48) SMN1; SMN2LMNAALDH1A1POLBMAPT
SCHEMBL17663880 0.83 HSP90AB1 (0.40) SMN1; SMN2LMNAALDH1A1TSHRCYP2C9
SCHEMBL27433056 0.81 MEN1 (0.66) SMN1; SMN2LMNAALDH1A1MEN1KMT2A
SCHEMBL17664019 0.74 ALDH1A1 (0.53) SMN1; SMN2LMNAALDH1A1TSHRPOLB
SCHEMBL17664014 0.74 PARP1 (0.38) SMN1; SMN2LMNAALDH1A1TSHRCYP2C9
SCHEMBL20448014 0.73 MAOB (0.50) SMN1; SMN2LMNAALDH1A1
SCHEMBL13500477 0.72 LMNA (0.51) SMN1; SMN2LMNAALDH1A1TSHRCYP2C9
SCHEMBL14880495 0.72 LTA4H (0.65) SMN1; SMN2LMNAALDH1A1TSHRMAPT
Ammonia Solution, Strong SCHEMBL29153964 0.71 PDE3B (0.58) SMN1; SMN2LMNAALDH1A1POLBPDE3B
SCHEMBL22912582 0.71 L3MBTL1 (0.41) SMN1; SMN2LMNAALDH1A1TSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed
WO-2016053855-A1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS THE SCRIPPS RESEARCH INSTITUTE (US) 2016-04-07 WO disclosed