SCHEMBL17665686

SCHEMBL17665686

Nc1ccccc1OC1c2ccccc2-n2cncc21

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.47
IDO1 P14902 2/20 0.42
ALDH1A1 P00352 1/20 0.32
ADRA2B P18089 1/20 0.32
PTGS1 P23219 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17651951 0.85 TDO2 (0.46) TDO2IDO1ALDH1A1
SCHEMBL17651954 0.85 TDO2 (0.46) TDO2IDO1
SCHEMBL17665684 0.84 TDO2 (0.46) TDO2IDO1
SCHEMBL17651968 0.82 TDO2 (0.43) TDO2IDO1
SCHEMBL17665692 0.82 TDO2 (0.52) TDO2IDO1
SCHEMBL17651987 0.81 TDO2 (0.50) TDO2IDO1
SCHEMBL17665352 0.81 TDO2 (0.47) TDO2IDO1
SCHEMBL17665351 0.79 TDO2 (0.48) TDO2IDO1
SCHEMBL17665691 0.79 SLC9A3 (0.43) TDO2ALDH1A1GPBAR1
SCHEMBL17665685 0.79 TDO2 (0.41) TDO2IDO1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016051181-A1 4H-IMIDAZO[1,5-A]INDOLE DERIVATIVES AND THEIR USE AS INDOLEAMINE 2,3-DIOXYGENASE (IDO) AND/OR TRYPTOPHAN 2,3-DIOXYGENASE (TD02) MODULATORS REDX PHARMA PLC (GB) 2016-04-07 WO disclosed