Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | CYP1A2 | P05177 | 2/20 | 0.52 |
| ▸ | GRM8 | O00222 | 1/20 | 0.52 |
| ▸ | GRM6 | O15303 | 1/20 | 0.52 |
| ▸ | GRIN2D | O15399 | 1/20 | 0.52 |
| ▸ | GRIN3B | O60391 | 1/20 | 0.52 |
| ▸ | GSR | P00390 | 1/20 | 0.52 |
| ▸ | GRIK1 | P39086 | 1/20 | 0.52 |
| ▸ | GRM5 | P41594 | 1/20 | 0.52 |
| ▸ | GRIA1 | P42261 | 1/20 | 0.52 |
| ▸ | GRIA2 | P42262 | 1/20 | 0.52 |
| ▸ | GRIA3 | P42263 | 1/20 | 0.52 |
| ▸ | SLC1A3 | P43003 | 1/20 | 0.52 |
| ▸ | SLC1A2 | P43004 | 1/20 | 0.52 |
| ▸ | SLC1A1 | P43005 | 1/20 | 0.52 |
| ▸ | GRIA4 | P48058 | 1/20 | 0.52 |
| ▸ | GRIN1 | Q05586 | 1/20 | 0.52 |
| ▸ | GRIN2A | Q12879 | 1/20 | 0.52 |
| ▸ | GRIK2 | Q13002 | 1/20 | 0.52 |
| ▸ | GRIK3 | Q13003 | 1/20 | 0.52 |
| ▸ | GRIN2B | Q13224 | 1/20 | 0.52 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Leucine SCHEMBL6130154 | 0.91 | SLC7A5 (0.51) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| SCHEMBL2482058 | 0.88 | ALOX15 (0.53) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| D-Glutamate SCHEMBL28632361 | 0.83 | SLC1A3 (0.46) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| SCHEMBL28554464 | 0.82 | SLC7A5 (0.40) | GRIK1GRIA1GRIA2SLC1A3SLC1A2 | |
| SCHEMBL4537589 | 0.82 | GABRP (0.54) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| SCHEMBL7780572 | 0.82 | GABRP (0.54) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| Asparagine SCHEMBL6130108 | 0.82 | ALOX15 (0.50) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| SCHEMBL3422700 | 0.81 | SLC1A2 (0.45) | GRIK1SLC1A3SLC1A2SLC1A1GRIK2 | |
| Cysteine SCHEMBL8071966 | 0.81 | ALOX15 (0.49) | CYP1A2GRM8GRM6GRIN2DGRIN3B | |
| SCHEMBL135879 | 0.80 | SLC7A5 (0.41) | SLC1A3SLC1A2SLC1A1SLC7A5 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2011053167-A1 | TRANSCRIPTION FACTOR POLYNUCLEOTIDES AND THEIR USE | GRASSLANZ TECHNOLOGY LIMITED (NZ) | 2011-05-05 | — | — | WO | claimed |
| EP-4010364-A1 | MODIFIED HUMAN VARIABLE DOMAINS | Merus N.V. (NL) | 2022-06-15 | — | — | EP | disclosed |
| WO-2021025555-A1 | MODIFIED HUMAN VARIABLE DOMAINS | MERUS N.V. (NL) | 2021-02-11 | — | — | WO | disclosed |
| EP-3772518-A1 | MODIFIED HUMAN VARIABLE DOMAINS | Merus N.V. (NL) | 2021-02-10 | — | — | EP | disclosed |
| US-8900849-B2 | Oxygen-regulated microorganisms | SCARAB GENOMICS, LLC (US) | 2014-12-02 | — | — | US | disclosed |
| US-20140186957-A1 | ENGINEERED TAL EFFECTOR PROTEINS WITH ENHANCED DNA TARGETING CAPACITY | FRED HUTCHINSON CANCER RESEARCH CENTER (US) | 2014-07-03 | — | — | US | disclosed |
| US-8354372-B2 | Cyclised alpha-conotoxin peptides | THE UNIVERSITY OF QUEENSLAND (AU) | 2013-01-15 | — | — | US | disclosed |
| WO-2011053167-A1 | TRANSCRIPTION FACTOR POLYNUCLEOTIDES AND THEIR USE | GRASSLANZ TECHNOLOGY LIMITED (NZ) | 2011-05-05 | — | — | WO | disclosed |
| US-20090053792-A1 | OXYGEN-REGULATED MICROORGANISMS | SCARAB GENOMICS, LLC (US) | 2009-02-26 | — | — | US | disclosed |