SCHEMBL17674396

SCHEMBL17674396

CCC(N)S(=N)(=O)c1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.44
PLCG1 P19174 1/20 0.42
CA12 O43570 3/20 0.40
CA9 Q16790 2/20 0.40
CA1 P00915 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
CA7 P43166 1/20 0.38
F2 P00734 2/20 0.37
PRSS1 P07477 2/20 0.37
PRSS2 P07478 2/20 0.37
PRSS3 P35030 2/20 0.37
SLC1A3 P43003 1/20 0.36
SLC1A2 P43004 1/20 0.36
SLC1A1 P43005 1/20 0.36
GAA P10253 3/20 0.36
MMP2 P08253 2/20 0.36
MMP1 P03956 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17674064 0.79 PLCG1 (0.42) CA2PLCG1CA12CA9CA1
SCHEMBL16124948 0.75 CA2 (0.46) CA2PLCG1CA12CA9CA1
SCHEMBL20590400 0.72 PLCG1 (0.52) CA2PLCG1CA12CA9CA1
SCHEMBL12674211 0.72 MMP2 (0.47) CA2PLCG1CA12CA9CA1
SCHEMBL17674087 0.72 MMP2 (0.44) CA2PLCG1CA12CA9CA1
SCHEMBL13813079 0.72 MMP2 (0.47) CA2PLCG1CA12CA9CA1
SCHEMBL9628601 0.68 CA2 (0.52) CA2PLCG1CA12CA9CA1
SCHEMBL24698628 0.68 CA2 (0.65) CA2PLCG1CA12CA9CA1
SCHEMBL5375 0.68 PLCG1 (0.70) CA2PLCG1CA12CA9CA1
SCHEMBL29025607 0.67 CA2 (0.56) CA2PLCG1CA12CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016054807-A1 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed