SCHEMBL17674698

SCHEMBL17674698

COc1cc(F)c(-c2c(C)nn(C)c2C(O)c2ccc(F)cc2F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.38
PDE10A Q9Y233 1/20 0.38
CYP1A2 P05177 2/20 0.38
GRM8 O00222 1/20 0.38
GRM7 Q14831 1/20 0.38
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 2/20 0.34
MAPK14 Q16539 1/20 0.34
APLNR P35414 1/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 2/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
PRKDC P78527 1/20 0.30
THRB P10828 1/20 0.30
CPS1 P31327 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15952664 0.86 CES2 (0.33) CYP1A2CYP3A4CYP2C9CYP2C19POLB
SCHEMBL170324 0.78 HSD11B1 (0.39) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL17674748 0.76 MAPK14 (0.41) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL17674744 0.75 MAPK14 (0.50) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL169795 0.74 PGR (0.36) CYP1A2CYP3A4CYP2C9CYP2C19POLB
SCHEMBL9998142 0.72 ADORA1 (0.41) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL17674735 0.72 CYP1A2 (0.39) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL17242927 0.71 MC4R (0.34) PDE2ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL15952683 0.71 PGR (0.31) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL15952778 0.71 IDO1 (0.32) MAPTKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055801-A2 AGRICULTURAL CHEMICALS REDAG CROP PROTECTION LTD (GB) 2016-04-14 WO disclosed
WO-2016055801-A2 AGRICULTURAL CHEMICALS REDAG CROP PROTECTION LTD (GB) 2016-04-14 WO disclosed