SCHEMBL17680425

SCHEMBL17680425

O=C(O)Cn1c(-c2ccns2)cc2cc(F)ccc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 2/20 0.48
NTRK3 Q16288 1/20 0.48
LMNA P02545 3/20 0.47
THRB P10828 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
TP53 P04637 3/20 0.45
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CCR2 P41597 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17680428 0.84 ALDH1A1 (0.53) NTRK1NTRK3LMNATHRBRXFP1
SCHEMBL17674413 0.81 KDM4E (0.43) NTRK1NTRK3LMNATHRBRXFP1
SCHEMBL17674247 0.80 NTRK1 (0.47) NTRK1LMNATHRBRXFP1TP53
SCHEMBL17680515 0.78 NTRK1 (0.45) NTRK1NTRK3LMNATHRBRXFP1
SCHEMBL17674262 0.77 NTRK1 (0.50) NTRK1LMNATHRBRXFP1TP53
SCHEMBL17680501 0.77 L3MBTL1 (0.71) NTRK1LMNATHRBRXFP1L3MBTL1
SCHEMBL17680316 0.76 NTRK1 (0.44) NTRK1LMNATHRBRXFP1TP53
SCHEMBL17674385 0.76 NTRK1 (0.45) NTRK1NTRK3LMNATHRBRXFP1
SCHEMBL17680320 0.76 NTRK1 (0.47) NTRK1LMNATHRBRXFP1TP53
SCHEMBL17674391 0.75 NTRK1 (0.60) NTRK1NTRK3LMNATHRBRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016054807-A1 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed