SCHEMBL17680474

SCHEMBL17680474

N=S(=O)(c1ccc(Br)cc1)C1CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.45
HTT P42858 2/20 0.44
MAPK1 P28482 1/20 0.44
PLCG1 P19174 1/20 0.43
MMP2 P08253 3/20 0.41
CA12 O43570 2/20 0.41
CA9 Q16790 1/20 0.41
CA1 P00915 1/20 0.41
MMP1 P03956 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP13 P45452 1/20 0.41
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSP90AA1 P07900 1/20 0.39
GAA P10253 2/20 0.39
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38
F2 P00734 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29850006 0.83 ALDH1A1 (0.48) CA2HTTMAPK1MMP2CA1
SCHEMBL17680275 0.82 CA2 (0.41) CA2HTTMAPK1PLCG1MMP2
SCHEMBL486801 0.80 HTR6 (0.46) CA2CA12CA9CA1ALDH1A1
SCHEMBL24008845 0.79 GAA (0.48) CA2MMP2CA12CA9CA1
SCHEMBL2412999 0.78 CA2 (0.48) CA2HTTMAPK1PLCG1MMP2
SCHEMBL29849710 0.76 MAOB (0.44) ALDH1A1SMN1; SMN2GAACDK1CDK2
SCHEMBL875209 0.75 CA1 (0.50) CA2HTTMMP2CA12CA9
SCHEMBL24010099 0.75 MMP13 (0.55) CA2HTTMMP2CA1MMP1
SCHEMBL24129786 0.75 CA2 (0.50) CA2ALDH1A1GAAF2LMNA
SCHEMBL883464 0.75 CA1 (0.50) CA2HTTMMP2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023104035-A1 SUBSTITUTED MONOCYCLIC OR BICYCLIC HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 英矽智能科技(上海)有限公司 2023-06-15 WO disclosed
WO-2016054807-A1 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed