SCHEMBL1768067

SCHEMBL1768067

CCCCC(C)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 5/20 0.47
ALDH1A1 P00352 1/20 0.45
CES1 P23141 4/20 0.45
MAOA P21397 8/20 0.43
MAOB P27338 8/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
CASP3 P42574 2/20 0.41
CAPN9 O14815 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9114249 0.94 TGM2 (0.45) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL1767901 0.91 TGM2 (0.50) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL5330038 0.84 TGM2 (0.53) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL1767975 0.82 TGM2 (0.42) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL4444879 0.79 TGM2 (0.55) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL1767899 0.76 TGM2 (0.44) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL3742475 0.74 MAOB (0.70) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL16111115 0.74 CES1 (0.53) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL17274920 0.73 ALDH1A1 (0.53) TGM2ALDH1A1CES1MAOAMAOB
SCHEMBL19674436 0.73 TBXAS1 (0.54) ALDH1A1MAOAMAOBPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed