SCHEMBL17680903

SCHEMBL17680903

O=C1CCNc2c(cccc2C(=O)OCc2ccccc2)N1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 3/20 0.64
BRD4 O60885 2/20 0.64
ALDH1A1 P00352 3/20 0.48
TDP1 Q9NUW8 3/20 0.47
MAPK1 P28482 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 1/20 0.46
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
POLB P06746 1/20 0.44
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
MMP12 P39900 2/20 0.43
MMP1 P03956 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.42
TSHR P16473 2/20 0.42
CYP3A4 P08684 1/20 0.42
CASP3 P42574 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22369307 0.87 BRD4 (0.54) CREBBPBRD4ALDH1A1TDP1MAPK1
SCHEMBL17673280 0.78 CREBBP (1.00) CREBBPBRD4
SCHEMBL22368749 0.78 BRD4 (0.61) CREBBPBRD4ALDH1A1TDP1MAPK1
SCHEMBL21027971 0.74 BRD4 (0.56) CREBBPBRD4ALDH1A1TDP1MAPK1
SCHEMBL22368804 0.74 CREBBP (0.62) CREBBPBRD4ALDH1A1
SCHEMBL17680672 0.74 CREBBP (0.64) CREBBPBRD4CRBNMAOAMAOB
SCHEMBL17680982 0.74 CREBBP (0.64) CREBBPBRD4ALDH1A1
SCHEMBL17680977 0.72 CREBBP (0.68) CREBBPBRD4ALDH1A1TSHR
SCHEMBL22368660 0.72 CREBBP (0.60) CREBBPBRD4NPC1DDB1CRBN
SCHEMBL50441 0.71 ALDH1A1 (0.89) ALDH1A1TDP1MAPK1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055028-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2016-04-14 WO disclosed