SCHEMBL17715580

SCHEMBL17715580

C/N=C1\NC(C)(CC(C)C)C(=O)N1CCC1CCN(C(=O)c2cccc(OC)c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.47
HSD11B1 P28845 2/20 0.44
MGLL Q99685 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 3/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520759 0.89 LMNA (0.49) LMNAHSD11B1MGLLL3MBTL1ALDH1A1
SCHEMBL7520594 0.82 LMNA (0.48) LMNAHSD11B1MGLLL3MBTL1ALDH1A1
SCHEMBL13723607 0.80 SMN1; SMN2 (0.35) LMNAALDH1A1KMT2A
SCHEMBL7520771 0.78 POLB (0.43) LMNAHSD11B1MGLLALDH1A1DRD2
SCHEMBL13722650 0.78 SMN1; SMN2 (0.43) HTTKMT2A
SCHEMBL7521184 0.76 HDAC3 (0.42) ALDH1A1DRD2HPGDTSHRHTT
SCHEMBL7520491 0.75 HTT (0.43) LMNAMGLLHTTMEN1KMT2A
SCHEMBL7522027 0.75 LMNA (0.46) LMNAHSD11B1ALDH1A1TP53HPGD
SCHEMBL8825345 0.75 ACHE (0.56) LMNAHSD11B1MGLLL3MBTL1ALDH1A1
SCHEMBL7523356 0.74 MGLL (0.47) LMNAHSD11B1MGLLALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097387-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2016-05-04 EP disclosed