SCHEMBL17734616

SCHEMBL17734616

Cc1cc(N(c2cccc(-c3ccccc3)c2)c2ccccc2C)ccc1-c1ccc(N(c2cccc(-c3ccccc3)c2)c2ccccc2C)cc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.37
TYMS P04818 1/20 0.33
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
TNKS2 Q9H2K2 1/20 0.32
MGLL Q99685 1/20 0.32
KDM4E B2RXH2 1/20 0.31
SLC6A9 P48067 1/20 0.31
MAOA P21397 2/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
HTR7 P34969 1/20 0.31
MAOB P27338 1/20 0.30
HSD17B1 P14061 1/20 0.30
HSD17B2 P37059 1/20 0.30
MEN1 O00255 1/20 0.30
APAF1 O14727 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17734613 0.91 ESR2 (0.39) ESR2TYMSCA12CA1CA2
SCHEMBL19844330 0.91 MGLL (0.37) TYMSTNKS2MGLLMAOAMAOB
SCHEMBL17734608 0.90 ESR2 (0.39) ESR2TYMSCA12CA1CA2
SCHEMBL22182144 0.89 TNKS2 (0.37) TYMSTNKS2MGLLKDM4EMAOA
SCHEMBL1702664 0.89 CYP3A4 (0.35) ESR2KDM4EHSD17B1HSD17B2MEN1
SCHEMBL19393523 0.88 TNKS2 (0.36) TYMSTNKS2MGLLKDM4EMAOA
SCHEMBL17734761 0.86 TYMS (0.34) TYMSTNKS2MGLLMAOAMAOB
SCHEMBL11321702 0.84 HSD17B1 (0.36) HSD17B1HSD17B2MEN1APAF1NPC1
SCHEMBL11330069 0.84 HSD17B1 (0.35) ESR2HSD17B1HSD17B2LMNA
SCHEMBL14179892 0.83 HSD17B1 (0.41) ESR2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160133847-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT IDEMITSU KOSAN CO., LTD. (JP) 2016-05-12 US disclosed
US-20160133847-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT IDEMITSU KOSAN CO., LTD. (JP) 2016-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160133847-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT ARL1, CCNL2, APOL1 ESR2 9/4885TYMS 4657/4885CA12 3357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.