SCHEMBL17737239

SCHEMBL17737239

O=C(O)c1ccccc1Cc1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.67
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
FOLH1 Q04609 1/20 0.53
PTPN1 P18031 5/20 0.48
ALDH1A1 P00352 3/20 0.46
MAPK1 P28482 1/20 0.46
GAA P10253 1/20 0.46
PTPN2 P17706 1/20 0.46
PTPN6 P29350 1/20 0.46
ALOX15 P16050 1/20 0.45
CYP2C9 P11712 1/20 0.44
HIF1A Q16665 1/20 0.44
KDM6B O15054 1/20 0.44
ALKBH2 Q6NS38 1/20 0.44
ALKBH3 Q96Q83 1/20 0.44
FTO Q9C0B1 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
KDM2A Q9Y2K7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23003 0.87 TSHR (0.79) TSHRCA1CA2CA9FOLH1
SCHEMBL28370887 0.85 TSHR (0.76) TSHRCA1CA2CA9FOLH1
Ammonia Solution, Strong SCHEMBL27527756 0.85 TSHR (0.76) TSHRCA1CA2CA9FOLH1
SCHEMBL29373730 0.84 KDR (0.57) TSHRFOLH1ALDH1A1GAAKDM6B
SCHEMBL1161694 0.84 CDC7 (0.50) TSHRCA1CA2CA9ALDH1A1
SCHEMBL9368471 0.84 TSHR (0.47) TSHRCA1CA2CA9ALDH1A1
SCHEMBL9621815 0.82 TSHR (0.45) TSHRCA1CA2CA9ALDH1A1
Ethylene Glycol SCHEMBL1817402 0.81 TSHR (0.71) TSHRCA1CA2CA9FOLH1
Acetic Acid SCHEMBL28245857 0.81 TSHR (0.71) TSHRCA1CA2CA9FOLH1
SCHEMBL258224 0.81 KDM6B (0.59) TSHRPTPN1ALDH1A1PTPN2PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9638690-B2 Compounds and compositions for use as alkylating agent sensors and methods of use thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-05-02 US disclosed
US-9638690-B2 Compounds and compositions for use as alkylating agent sensors and methods of use thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-05-02 US disclosed
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-05-12 US disclosed
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-05-12 US disclosed
CN-101384183-B Compounds comprising linked heteroaryl moieties and their use as novel umami flavor modifiers, tastants and taste enhancers for comestible compositions SENOMYX INC 2012-07-04 CN disclosed
CN-101384183-A Compounds comprising linked heteroaryl moieties and their use as novel umami flavor modifiers, tastants and taste enhancers for comestible compositions SENOMYX INC (US) 2009-03-11 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160131641-A1 COMPOUNDS AND COMPOSITIONS FOR USE AS ALKYLATING AGENT SENSORS AND METHODS OF USE THEREOF MGMT, MCL1, OGG1 TSHR 3834/4885CA1 219/4885CA2 478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.