SCHEMBL17758477

SCHEMBL17758477

CCc1cc(C(=O)NCCN(C)C)ccc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
TLR9 Q9NR96 2/20 0.58
TLR8 Q9NR97 2/20 0.58
TLR7 Q9NYK1 2/20 0.58
ALDH1A1 P00352 2/20 0.56
TP53 P04637 1/20 0.52
KIFC1 Q9BW19 1/20 0.52
KMT2A Q03164 4/20 0.51
MEN1 O00255 2/20 0.51
USP2 O75604 1/20 0.51
DRD2 P14416 1/20 0.50
DRD3 P35462 1/20 0.50
HRH3 Q9Y5N1 1/20 0.50
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MCHR1 Q99705 1/20 0.49
PRMT5 O14744 1/20 0.49
WDR77 Q9BQA1 1/20 0.49
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17758484 0.86 ROCK2 (0.61) TMEM97SIGMAR1ALDH1A1TP53KMT2A
SCHEMBL19657230 0.85 TMEM97 (0.56) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL17758471 0.85 SMPD1 (0.63) TMEM97SIGMAR1TLR8TLR7ALDH1A1
SCHEMBL17676475 0.83 LMNA (0.54) TMEM97SIGMAR1ALDH1A1TP53KMT2A
SCHEMBL20094150 0.82 SMN1; SMN2 (0.55) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL20682518 0.82 TMEM97 (0.53) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL19651848 0.82 ALDH1A1 (0.53) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL15656703 0.81 ALDH1A1 (0.52) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL1559022 0.81 ALDH1A1 (0.52) TMEM97SIGMAR1TLR9TLR8TLR7
SCHEMBL13575527 0.81 ALDH1A1 (0.55) TLR9TLR8TLR7ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016077378-A1 SUBSTITUTED PYRROLOPYRDINES AS INHIBITORS OF BROMODOMAIN GENENTECH, INC. (US) 2016-05-19 WO disclosed