SCHEMBL17758484

SCHEMBL17758484

CCCNC(=O)c1ccc(OC)c(CC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.61
TP53 P04637 1/20 0.57
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
SMPD1 P17405 1/20 0.54
TMEM97 Q5BJF2 1/20 0.53
SIGMAR1 Q99720 1/20 0.53
POLB P06746 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPT P10636 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
HDAC3 O15379 1/20 0.51
HDAC2 Q92769 1/20 0.51
HPGD P15428 2/20 0.50
ALDH1A1 P00352 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17758471 0.90 SMPD1 (0.63) ROCK2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL17676475 0.88 LMNA (0.54) TP53NPC1RAB9ATMEM97SIGMAR1
SCHEMBL930908 0.88 ROCK2 (0.76) ROCK2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL17758477 0.86 TMEM97 (0.58) TP53NPC1RAB9ASMN1; SMN2TMEM97
SCHEMBL14340547 0.85 TAS1R3 (0.64) ROCK2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL24021265 0.85 POLB (0.70) TP53NPC1RAB9ASMN1; SMN2SMPD1
SCHEMBL24021268 0.84 TLR7 (0.61) ROCK2TP53NPC1RAB9ASMPD1
SCHEMBL8324748 0.84 TAS1R3 (0.64) ROCK2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL8324517 0.84 TAS1R3 (0.65) ROCK2TP53NPC1RAB9ASMN1; SMN2
SCHEMBL17758615 0.83 SLC6A2 (0.56) TP53SMPD1MEN1KMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016077378-A1 SUBSTITUTED PYRROLOPYRDINES AS INHIBITORS OF BROMODOMAIN GENENTECH, INC. (US) 2016-05-19 WO disclosed