SCHEMBL17771973

SCHEMBL17771973

Cc1cc(C(=O)NCCCN(CCCN)CCS(=O)(=O)O)cc(C)c1OC(=O)c1c2ccccc2[n+](CCCS(=O)(=O)O)c2ccccc12

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
HDAC3 O15379 1/20 0.31
HTT P42858 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
FLT3 P36888 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16142712 0.95 DRD2 (0.33) DRD2DRD4DRD3HDAC3HTT
SCHEMBL18531453 0.89 LMNA (0.33) DRD2DRD4DRD3HDAC3HTT
SCHEMBL18531414 0.87 LMNA (0.33) DRD2DRD4DRD3HDAC3HTT
SCHEMBL17771978 0.86 SMN1; SMN2 (0.38) HTTKDM4EALDH1A1HPGD
SCHEMBL16142548 0.86 GRIN1 (0.33) GRIN1GRIN2AGRIN2BHDAC3FLT3
SCHEMBL16142686 0.86 GRIN1 (0.32) GRIN1GRIN2AGRIN2BHDAC3
SCHEMBL18531451 0.84 FLT3 (0.31) FLT3
SCHEMBL18531452 0.83 BCHE (0.30)
SCHEMBL17771976 0.82 SIGMAR1 (0.34) HTT
SCHEMBL18531415 0.81 BCHE (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3067345-A1 ZWITTERION-CONTAINING ACRIDINIUM COMPOUNDS Siemens Healthcare Diagnostics Inc. (US) 2016-09-14 EP disclosed
EP-2501681-B1 ZWITTERION-CONTAINING ACRIDINIUM COMPOUNDS SIEMENS HEALTHCARE DIAGNOSTICS (US) 2016-05-25 EP disclosed