SCHEMBL17778484

SCHEMBL17778484

CCc1cnc(I)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
PARP1 P09874 1/20 0.33
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
RAPGEF4 Q8WZA2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10310085 0.77 NOS3 (0.38) NOS3NOS1NOS2PARP1KDM4E
SCHEMBL19831176 0.77 RXRA (0.32) NOS3NOS1NOS2PARP1KDM4E
SCHEMBL25759811 0.76 NOS3 (0.36) NOS3NOS1NOS2PARP1KDM4E
SCHEMBL9128305 0.74 NOS3 (0.35) NOS3NOS1NOS2PARP1KDM4E
SCHEMBL10268101 0.74 NOS3 (0.56) NOS3NOS1NOS2PARP1
SCHEMBL9970964 0.74 NOS3 (0.35) NOS3NOS1NOS2PARP1KDM4E
SCHEMBL2597202 0.74 NOS3 (0.35) NOS3NOS1NOS2PARP1
SCHEMBL8631001 0.74 PTGS2 (0.36) NOS3NOS1NOS2RAPGEF4
SCHEMBL23626192 0.72
SCHEMBL2714235 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170073460-A1 POLYETHER KETONE COMPOUND AJINOMOTO CO., INC. (JP) 2017-03-16 US disclosed
WO-2016079712-A1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-26 WO disclosed