SCHEMBL17782894

SCHEMBL17782894

COC(=O)CNC(=O)Nc1ccc(OC)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
NPC1 O15118 3/20 0.68
CA12 O43570 1/20 0.64
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64
CA9 Q16790 1/20 0.64
SAE1 Q9UBE0 1/20 0.61
UBA2 Q9UBT2 1/20 0.61
ALDH1A1 P00352 1/20 0.59
HTT P42858 1/20 0.59
CYP1A2 P05177 1/20 0.57
CYP2C19 P33261 1/20 0.57
KDM4E B2RXH2 2/20 0.57
MEN1 O00255 2/20 0.57
MAPT P10636 2/20 0.57
KMT2A Q03164 2/20 0.57
PKM P14618 1/20 0.56
POLB P06746 1/20 0.56
FPR2 P25090 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1514347 0.87 RAB9A (0.68) RAB9ASMN1; SMN2NPC1SAE1UBA2
SCHEMBL5352692 0.83 LMNA (0.65) RAB9ASMN1; SMN2NPC1CA12CA1
SCHEMBL9435964 0.83 RAB9A (0.72) RAB9ASMN1; SMN2NPC1SAE1UBA2
SCHEMBL11092496 0.82 RAB9A (1.00) RAB9ASMN1; SMN2NPC1CA12CA1
SCHEMBL4588526 0.81 RAB9A (0.70) RAB9ASMN1; SMN2NPC1SAE1UBA2
SCHEMBL10633474 0.81 CA12 (0.65) RAB9ASMN1; SMN2NPC1CA12CA1
SCHEMBL8577837 0.80 SMN1; SMN2 (0.68) RAB9ASMN1; SMN2NPC1CA12CA1
SCHEMBL20708118 0.80 SMN1; SMN2 (0.68) RAB9ASMN1; SMN2NPC1SAE1UBA2
SCHEMBL17916794 0.80 SMN1; SMN2 (0.88) RAB9ASMN1; SMN2NPC1SAE1UBA2
Trifluoroacetic Acid SCHEMBL2891081 0.80 NPC1 (0.54) RAB9ASMN1; SMN2NPC1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9662328-B2 Targeting human thymidylate kinase induces DNA repair toxicity in malignant tumor cells NATIONAL TAIWAN UNIVERSITY (TW) 2017-05-30 US disclosed
US-20160151362-A1 TARGETING HUMAN THYMIDYLATE KINASE INDUCES DNA REPAIR TOXICITY IN MALIGNANT TUMOR CELLS NATIONAL TAIWAN UNIVERSITY (TW) 2016-06-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160151362-A1 TARGETING HUMAN THYMIDYLATE KINASE INDUCES DNA REPAIR TOXICITY IN MALIGNANT TUMOR CELLS DTYMK, TYMP, TK1 RAB9A 3942/4885SMN1; SMN2 4349/4885NPC1 4369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.