SCHEMBL17801072

SCHEMBL17801072

CS(=O)(=O)Nc1cccc(-c2n[nH]c3ccc(-c4nc(C5CCCN5)n[nH]4)cc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.46
AAK1 Q2M2I8 1/20 0.45
MAP2K4 P45985 2/20 0.41
MAP3K5 Q99683 1/20 0.41
NTRK1 P04629 1/20 0.41
TTK P33981 2/20 0.41
MAP2K7 O14733 1/20 0.41
AURKB Q96GD4 5/20 0.40
CLK4 Q9HAZ1 3/20 0.40
CDC7 O00311 1/20 0.40
PLK4 O00444 1/20 0.40
DAPK3 O43293 1/20 0.40
DYRK3 O43781 1/20 0.40
JAK2 O60674 1/20 0.40
ROCK2 O75116 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
CDK1 P06493 1/20 0.40
ROS1 P08922 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17801075 0.87 PDPK1 (0.52) MAP2K4MAP3K5TTKMAP2K7PLK4
SCHEMBL17801079 0.84 PDPK1 (0.49) AAK1CLK2CSNK2A1DYRK1AITK
SCHEMBL17801078 0.81 CSNK1D (0.49) CSNK1DMAP2K4MAP3K5TTKMAPK1
SCHEMBL17801071 0.79 MAP3K5 (0.54) MAP3K5DYRK1A
SCHEMBL17801077 0.75 PARP1 (0.43) MAP2K4MAP3K5AURKBMAP4K4CLK2
SCHEMBL8253362 0.74 CSNK1D (0.52) CSNK1DAAK1MAP2K4MAP3K5NTRK1
SCHEMBL5377458 0.71 CSNK1D (0.55) CSNK1DAAK1MAP2K4MAP3K5NTRK1
SCHEMBL17801093 0.69 CPT1A (0.63) CSNK1DAAK1
SCHEMBL17801086 0.68 PDPK1 (0.47) AAK1CLK2CSNK2A1DYRK1AITK
SCHEMBL1460755 0.68 MAPK1 (0.61) CSNK1DMAP2K4NTRK1TTKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed