SCHEMBL17816181

SCHEMBL17816181

O=C(O)CC1CCC(Sc2cc(C(=O)Nc3cc(F)c(F)c(F)c3)ccc2I)C1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 7/20 0.34
ITGB3 P05106 5/20 0.34
ITGA2B P08514 5/20 0.34
SOAT1 P35610 1/20 0.34
RARA P10276 2/20 0.34
RARB P10826 2/20 0.34
RARG P13631 2/20 0.34
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
KDM1A O60341 3/20 0.32
RCOR1 Q9UKL0 1/20 0.32
MAOA P21397 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17816184 0.91 NPC1 (0.42) DGAT1ITGB3ITGA2BSOAT1MAOA
SCHEMBL17784015 0.91 DGAT1 (0.37) DGAT1ITGB3ITGA2BSOAT1RARA
SCHEMBL17816187 0.87 NPC1 (0.45) DGAT1MAOATP53MAPTMAOB
SCHEMBL17816135 0.85 RARA (0.35) DGAT1RARARARBRARGKDM1A
SCHEMBL21991658 0.85 DGAT1 (0.40) DGAT1ITGB3ITGA2BSOAT1RARA
SCHEMBL17792189 0.85 DGAT1 (0.40) DGAT1ITGB3ITGA2BSOAT1RARA
SCHEMBL17784130 0.83 NPC1 (0.45) DGAT1ITGB3ITGA2BSOAT1MAOA
SCHEMBL17816156 0.83 RARA (0.36) DGAT1SOAT1RARARARBRARG
SCHEMBL17816078 0.83 RARA (0.36) DGAT1SOAT1RARARARBRARG
SCHEMBL17816134 0.83 RARA (0.36) DGAT1SOAT1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089990-A1 SULFIDE ALKYL AND PYRIDYL REVERSE SULFONAMIDE COMPOUNDS FOR HBV TREATMENT NOVIRA THERAPEUTICS, INC. (US) 2016-06-09 WO disclosed