SCHEMBL17826231

SCHEMBL17826231

CC(=O)Nc1ccc(C(C)=O)cc1-c1nnn[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
PRKCI P41743 1/20 0.37
TP53 P04637 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
MAPT P10636 3/20 0.36
KCNJ1 P48048 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA3 P0DMS8 2/20 0.35
NEU3 Q9UQ49 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.34
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
S100A4 P26447 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12434678 0.88 ALDH1A1 (0.40) ALDH1A1HDAC1HDAC6MAPTNPC1
SCHEMBL13973892 0.87 ALDH1A1 (0.40) ALDH1A1TP53HDAC1HDAC6MAPT
SCHEMBL12892206 0.80 ALDH1A1 (0.57) ALDH1A1NPC1RAB9AKDM4EHSD17B10
SCHEMBL11386472 0.80 PKM (0.41) ALDH1A1MAPTKCNJ1NPC1RAB9A
SCHEMBL6258779 0.78 CSF1R (0.34) ALDH1A1
SCHEMBL1463081 0.76 MEN1 (0.47) ALDH1A1TP53MAPTNPC1RAB9A
SCHEMBL1462966 0.74 MEN1 (0.54) ALDH1A1TP53MAPTNPC1RAB9A
SCHEMBL6710112 0.72 MAP3K5 (0.45) TP53HDAC1MAPTNPC1RAB9A
SCHEMBL7432657 0.71 XDH (0.51) TP53MAPTKCNJ1NPC1RAB9A
SCHEMBL1462306 0.71 IDH1 (0.48) TP53MAPTNPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9365612-B2 Caspase inhibitors UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2016-06-14 US disclosed