SCHEMBL17826574

SCHEMBL17826574

COc1ccccc1C(=O)NC(=S)Nc1ccc(NC(=O)CCCCN)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.63
CA2 P00918 2/20 0.63
CA9 Q16790 2/20 0.63
ALDH1A1 P00352 4/20 0.58
MAPT P10636 3/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TP53 P04637 1/20 0.58
SIRT2 Q8IXJ6 4/20 0.57
RAB9A P51151 2/20 0.53
GAA P10253 1/20 0.53
POLB P06746 1/20 0.52
HDAC3 O15379 2/20 0.52
HDAC1 Q13547 2/20 0.52
MAPK1 P28482 1/20 0.52
S1PR1 P21453 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1707492 0.86 SIRT2 (0.76) SIRT2
SCHEMBL17826593 0.85 SIRT2 (0.76) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL17826594 0.83 ALDH1A1 (0.64) CA1CA2CA9ALDH1A1KMT2A
SCHEMBL25132677 0.82 CA1 (0.67) CA1CA2CA9ALDH1A1MAPT
Hydrochloric Acid SCHEMBL3716563 0.80 CA1 (0.72) CA1CA2CA9ALDH1A1MAPT
SCHEMBL17826576 0.80 POLB (0.64) CA1CA2CA9ALDH1A1SMN1; SMN2
SCHEMBL17826586 0.80 SIRT2 (0.77) CA1CA2CA9ALDH1A1MAPT
SCHEMBL14096570 0.80 CA1 (0.72) CA1CA2CA9ALDH1A1MAPT
SCHEMBL14096549 0.80 RAB9A (0.74) CA1CA2CA9ALDH1A1MAPT
SCHEMBL14096572 0.79 MAPT (0.68) CA1CA2CA9ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9365508-B2 Aroyl thiourea derivatives UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2016-06-14 US disclosed