SCHEMBL17826752

SCHEMBL17826752

O=C(C1NC(c2cc(Cl)c(O)c(Cl)c2)=NO1)N(Cc1cccnc1)Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 1/20 0.41
NR1H3 Q13133 1/20 0.41
PKM P14618 1/20 0.38
UBE2M P61081 5/20 0.38
DCUN1D1 Q96GG9 5/20 0.38
NAMPT P43490 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
PLA2G1B P04054 1/20 0.37
HPGD P15428 1/20 0.37
VNN1 O95497 1/20 0.36
CHRM5 P08912 1/20 0.35
GRIN2B Q13224 2/20 0.35
POLB P06746 1/20 0.35
GRIN1 Q05586 1/20 0.35
PTGES O14684 1/20 0.35
AKR1C3 P42330 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17826743 0.90 NR1D1 (0.41) NR1D1NR1H3PKMUBE2MDCUN1D1
SCHEMBL1114708 0.75 NR1D1 (0.42) NR1D1NR1H3PKMUBE2MDCUN1D1
SCHEMBL3242548 0.75 SMN1; SMN2 (0.49) NR1D1NR1H3NAMPTVNN1GPBAR1
SCHEMBL2396944 0.70 GRIN2B (0.40) NR1D1NR1H3PKMUBE2MDCUN1D1
SCHEMBL1114600 0.66 CASP3 (0.44)
SCHEMBL1114301 0.65 SMN1; SMN2 (0.49) NR1D1NR1H3NAMPTVNN1GPBAR1
SCHEMBL8390987 0.64 HDAC1 (0.43) KMT2A
SCHEMBL1114279 0.63 MAPT (0.43) LMNAPOLB
SCHEMBL28977515 0.63 VNN1 (0.54) NR1D1NR1H3NAMPTMEN1KMT2A
SCHEMBL3235226 0.63 SCD5 (0.57) MEN1KMT2ALMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-B1 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES PATH DRUG SOLUTIONS (US) 2016-06-15 EP disclosed