SCHEMBL17833757

SCHEMBL17833757

Cc1cc2c(cc1CO)C(CSc1nnnn1-c1ccccc1)N(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.42
TSHR P16473 3/20 0.42
APOBEC3A P31941 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
LMNA P02545 1/20 0.41
POLB P06746 3/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NTRK1 P04629 1/20 0.38
NTRK2 Q16620 1/20 0.38
NFE2 Q16621 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17833751 0.84 GHSR (0.36) ALDH1A1LMNAMEN1MAPTKMT2A
SCHEMBL20705812 0.82 MTNR1B (0.45) ALDH1A1LMNAMEN1MAPTKMT2A
SCHEMBL17833755 0.77 MEN1 (0.41) LMNAMEN1KMT2A
SCHEMBL17833752 0.73 GHSR (0.41) ALDH1A1TSHRLMNAMEN1KMT2A
SCHEMBL17833754 0.73 GHSR (0.42)
SCHEMBL17821591 0.71 MTNR1B (0.49) ALDH1A1LMNAMEN1MAPTKMT2A
SCHEMBL17833756 0.69 GHSR (0.39) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL17821679 0.68 MTNR1B (0.46) LMNAMEN1KMT2A
SCHEMBL17864820 0.67 MTNR1B (0.45) MEN1MAPTKMT2A
SCHEMBL12295499 0.67 GHSR (0.39) LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170368051-A1 2-PHENETHENYLTETRAHYDRO ISOQUINOLINES USEFUL AS ANTI-HIV COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-12-28 US disclosed
US-9518022-B2 Anti-HIV compounds PROSETTA ANTIVIRAL INC. (US) 2016-12-13 US disclosed
US-20160168100-A1 ANTI-HIV COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160168100-A1 ANTI-HIV COMPOUNDS MAVS, SARS1, NFATC1 ALDH1A1 3741/4885TSHR 4858/4885APOBEC3A 419/4885
US-20170368051-A1 2-PHENETHENYLTETRAHYDRO ISOQUINOLINES USEFUL AS ANTI-HIV COMPOUNDS MAVS, EIF2AK2, POLRMT ALDH1A1 3748/4885TSHR 4860/4885APOBEC3A 712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.