SCHEMBL17835608

SCHEMBL17835608

CC(C)[Si](OCC[C@@H](O)c1ccccc1)(C(C)C)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.47
LMNA P02545 1/20 0.46
AOC3 Q16853 5/20 0.41
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DHFR P00374 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19666973 1.00 RIPK1 (0.47) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL16756832 0.83 SLC6A2 (0.38) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL25419566 0.82 LMNA (0.48) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL17835547 0.82 LMNA (0.48) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL27094502 0.77 RIPK1 (0.53) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL1520904 0.77 RIPK1 (0.53) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL14758666 0.76 RIPK1 (0.55) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL1779384 0.76 RIPK1 (0.55) RIPK1LMNAAOC3ALDH1A1KDM4E
SCHEMBL11228716 0.75 RIPK1 (0.53) RIPK1LMNAAOC3KDM4EL3MBTL1
SCHEMBL28428630 0.72 KMT2A (0.35) LMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10130619-B2 Amido thiadiazole derivatives as NADPH oxidase inhibitors GENKYOTEX SUISSE SA (CH) 2018-11-20 US disclosed
US-20170348296-A1 AMIDO THIADIAZOLE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SUISSE SA (CH) 2017-12-07 US disclosed
EP-3034500-A1 Amido thiazole derivatives as NADPH oxidase inhibitors GENKYOTEX SA (CH) 2016-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170348296-A1 AMIDO THIADIAZOLE DERIVATIVES AS NADPH OXIDASE INHIBITORS NOX1, NOX5, CYBB RIPK1 3578/4885LMNA 4266/4885AOC3 111/4885
US-10130619-B2 Amido thiadiazole derivatives as NADPH oxidase inhibitors NOX1, NOX5, CYBB RIPK1 3578/4885LMNA 4266/4885AOC3 111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.