SCHEMBL17844769

SCHEMBL17844769

CC(C)(C)OC(=O)NOC(=O)CCCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
SIGMAR1 Q99720 3/20 0.48
TDP1 Q9NUW8 2/20 0.47
KMT2A Q03164 1/20 0.47
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
MAPK1 P28482 1/20 0.46
ADRA1A P35348 1/20 0.46
HDAC4 P56524 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30678936 0.96 ALOX5 (0.48) ADRB2ADRB1ADRB3SIGMAR1HDAC1
SCHEMBL3786555 0.92 TDP1 (0.50) SIGMAR1TDP1KMT2ACA12CA1
SCHEMBL27413860 0.88 CA1 (0.42) ADRB2ADRB1ADRB3SIGMAR1CA1
SCHEMBL10578604 0.84 HDAC1 (0.56) ADRB2ADRB1ADRB3SIGMAR1TDP1
SCHEMBL1948655 0.82 CA12 (0.50) ADRB2ADRB1ADRB3MAPK1SMN1; SMN2
SCHEMBL6942862 0.81 CA12 (0.46) SIGMAR1CA12CA1CA7CA14
SCHEMBL28327204 0.80 SYK (0.48) KMT2AMAPK1SMN1; SMN2CA12CA1
SCHEMBL7083503 0.80 HTT (0.55) MAPK1SMN1; SMN2POLBIDO1
SCHEMBL9196120 0.79 MAPT (0.56) ADRB2ADRB1ADRB3TDP1KMT2A
SCHEMBL7101278 0.79 CA2 (0.41) CA1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102448-B Phenylpyrazole derivatives as ROCK1 and ROCK2 inhibitor 百时美施贵宝公司 2018-03-06 CN disclosed
WO-2016095088-A1 ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed