SCHEMBL3786555

SCHEMBL3786555

CC(C)(C)OC(=O)NOC(=O)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA7 P43166 1/20 0.48
CA14 Q9ULX7 1/20 0.48
CTSK P43235 2/20 0.46
CTSS P25774 1/20 0.46
IDO1 P14902 1/20 0.46
AKT1 P31749 2/20 0.46
ALDH1A1 P00352 1/20 0.45
SIGMAR1 Q99720 3/20 0.45
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
ATM Q13315 1/20 0.44
KMT2A Q03164 1/20 0.43
ACE P12821 1/20 0.43
KEAP1 Q14145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844769 0.92 ADRB2 (0.49) TDP1CA12CA1CA7CA14
SCHEMBL30678936 0.90 ALOX5 (0.48) CA12CA1CA7CA14CTSK
SCHEMBL7101278 0.87 CA2 (0.41) CA1IDO1PPARGPPARA
SCHEMBL3901264 0.86 CA2 (0.40) CA12CA1CA7CA14AKT1
SCHEMBL6942862 0.86 CA12 (0.46) CA12CA1CA7CA14CTSK
SCHEMBL1948655 0.85 CA12 (0.50) CA12CA1CA7CA14CTSK
SCHEMBL9006857 0.84 TDP1 (0.56) TDP1CA12CA7CA14ALDH1A1
SCHEMBL1380801 0.82 TDP1 (0.61) TDP1ALDH1A1KMT2AKEAP1
SCHEMBL23467154 0.80 CA2 (0.45) CA12CA1CA7CA14KMT2A
SCHEMBL23859885 0.80 CA1 (0.37) CA12CA1CA7CA14CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109867630-A - 1 receptor modulators of novel glp-1 赛尔基因第二国际有限公司 2019-06-11 CN disclosed
CN-105593225-B novel GLP-1 receptor modulators 赛尔基因第二国际有限公司 2019-04-16 CN disclosed
EP-3353145-A1 PRODRUGS OF GAMMA-HYDROXYBUTYRIC ACID, COMPOSITIONS AND USES THEREOF XW Laboratories Inc. (KY) 2018-08-01 EP disclosed
WO-2017050259-A1 PRODRUGS OF GAMMA-HYDROXYBUTYRIC ACID, COMPOSITIONS AND USES THEREOF XW LABORATORIES INC. (KY) 2017-03-30 WO disclosed
WO-2017049470-A1 PRODRUGS OF GAMMA-HYDROXYBUTYRIC ACID, COMPOSITIONS AND USES THEREOF XW LABORATORIES INC. (CN) 2017-03-30 WO disclosed
WO-2010024762-A1 PREPARATION OF β-PHENYL-ISOSERINE DERIVATIVES ORGANOCLICK AKTIEBOLAG (SE) 2010-03-04 WO disclosed