SCHEMBL17846112

SCHEMBL17846112

CNc1ccccc1CCNC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.45
MTNR1B P49286 1/20 0.44
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HIF1A Q16665 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC16A3 O15427 1/20 0.40
POLB P06746 2/20 0.40
ITGB3 P05106 1/20 0.40
ITGAV P06756 1/20 0.40
PTGS2 P35354 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845992 0.89 KMT2A (0.49) TMEM97SIGMAR1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL17846142 0.87 SLC16A3 (0.48) TMEM97SIGMAR1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL29157005 0.85 TMEM97 (0.55) MTNR1AMTNR1BTMEM97SIGMAR1HIF1A
SCHEMBL17258879 0.82 ALDH1A1 (0.49) TMEM97SIGMAR1NPC1RAB9AL3MBTL1
SCHEMBL20564338 0.81 MTNR1A (0.44) MTNR1AMTNR1BL3MBTL1ALDH1A1MAPT
SCHEMBL10348018 0.80 ALDH1A1 (0.54) MTNR1AMTNR1BALDH1A1KMT2AMAPT
SCHEMBL3822300 0.80 L3MBTL1 (0.42) MTNR1AMTNR1BL3MBTL1ALDH1A1KMT2A
SCHEMBL11263494 0.79 KEAP1 (0.48) L3MBTL1ALDH1A1SMN1; SMN2POLBITGB3
SCHEMBL20563681 0.78 HPGD (0.47) MTNR1AMTNR1BNPC1RAB9AALDH1A1
SCHEMBL5671835 0.77 MTNR1A (0.57) MTNR1AMTNR1BNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233859-A1 ERK INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-10-25 EP disclosed
WO-2016100051-A1 ERK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed