SCHEMBL17848468

SCHEMBL17848468

Cc1cccc(OCCN2CCC(Oc3cccnc3)C2)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
DRD2 P14416 4/20 0.46
DRD3 P35462 4/20 0.46
KDM4E B2RXH2 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
PDE10A Q9Y233 1/20 0.44
KDM1A O60341 1/20 0.44
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6311368 0.78 CHRNB2 (0.49) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL21620973 0.76 LTA4H (0.58) HTR1AHTR7KDM4EL3MBTL1KMT2A
SCHEMBL12642591 0.76 CHRNB2 (0.57) CHRNB2CHRNA4DRD2DRD3KDM1A
SCHEMBL24521960 0.75 CHRNB2 (0.54) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL6311327 0.75 CHRNB2 (0.54) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL6306245 0.75 CHRNB2 (0.54) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL7237136 0.73 CHRNB2 (0.55) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL7530388 0.73 CHRNB2 (0.55) CHRNB2CHRNA4PDE3BPDE3APDE10A
SCHEMBL14426319 0.71 KDM4E (0.78) HTR1AHTR7KDM4EL3MBTL1KMT2A
SCHEMBL10262282 0.71 SLC6A2 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed