SCHEMBL17848964

SCHEMBL17848964

COc1ccc2nc(SC(C)C)cnc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 6/20 0.48
PDGFRA P16234 6/20 0.48
POLB P06746 3/20 0.47
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
MEN1 O00255 2/20 0.47
RAB9A P51151 2/20 0.47
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
NQO2 P16083 1/20 0.47
HPGDS O60760 6/20 0.43
EGFR P00533 2/20 0.43
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
F2 P00734 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29991269 0.76 ALDH1A1 (0.51) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL20595475 0.76 ALDH1A1 (0.51) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL557973 0.76 NCF1 (0.59) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL29991874 0.74 ALDH1A1 (0.56) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL28035890 0.74 RAB9A (0.56) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL621880 0.74 ALDH1A1 (0.56) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL558148 0.72 ALDH1A1 (0.55) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL13666129 0.72 ALDH1A1 (0.55) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL31033500 0.72 ALDH1A1 (0.55) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2
SCHEMBL10214298 0.70 MEN1 (0.87) PDGFRBPDGFRAPOLBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100101-A1 RUTHENIUM-BASED METATHESIS PRE-CATALYST COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed