SCHEMBL17849205

SCHEMBL17849205

N=C(c1ccc(C(N)=O)c(F)c1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.32
MAPK14 Q16539 1/20 0.31
MAP2K2 P36507 1/20 0.31
MAP2K1 Q02750 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GUSB P08236 1/20 0.31
F10 P00742 1/20 0.31
PIM1 P11309 1/20 0.31
BAD Q92934 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
JAK1 P23458 2/20 0.30
JAK3 P52333 2/20 0.30
JAK2 O60674 1/20 0.30
AURKA O14965 1/20 0.30
RPS6KB1 P23443 1/20 0.30
MAPK7 Q13164 1/20 0.30
MAPK8 P45983 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623554 0.89 MAPK14 (0.33) DGAT1MAPK14MAP2K2MAP2K1ALDH1A1
SCHEMBL17849237 0.86 RORC (0.33) MAPK14ALDH1A1GUSB
SCHEMBL17849236 0.86 RORC (0.36) MAPK14MAP2K1PKMMAPK7
SCHEMBL16726665 0.83 ALDH2 (0.33)
SCHEMBL16623544 0.82 MEN1 (0.32) MAPK14MAPK8
SCHEMBL16623547 0.80 SYK (0.36) ALDH1A1
SCHEMBL16623468 0.79 MPO (0.31) MAPK8
SCHEMBL17849215 0.78 CRBN (0.38)
SCHEMBL17849213 0.78 POLB (0.35) L3MBTL1
SCHEMBL17849202 0.78 SMN1; SMN2 (0.44) ALDH1A1L3MBTL1MAPK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed