SCHEMBL17849236

SCHEMBL17849236

N=C(c1cc(F)cc(C(N)=O)c1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.36
PARP1 P09874 1/20 0.35
MAPK7 Q13164 4/20 0.33
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
GAA P10253 2/20 0.32
MAPK14 Q16539 1/20 0.32
LMNA P02545 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31
MAP2K1 Q02750 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849237 0.86 RORC (0.33) RORCPARP1MAPK14
SCHEMBL17849205 0.86 DGAT1 (0.32) MAPK7MAPK14PKMMAP2K1
SCHEMBL16623544 0.84 MEN1 (0.32) MAPK14KMT2A
SCHEMBL16726665 0.82 ALDH2 (0.33) ITGB2ICAM1ITGALKMT2A
SCHEMBL16623603 0.81 PARP1 (0.36) RORCPARP1MAP2K1
SCHEMBL16623468 0.81 MPO (0.31)
SCHEMBL16623547 0.80 SYK (0.36)
SCHEMBL17849215 0.78 CRBN (0.38)
SCHEMBL16726696 0.77 HDAC6 (0.41) RORCLMNA
SCHEMBL18052610 0.77 MAPK10 (0.41) MAPK7MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed