SCHEMBL17849237

SCHEMBL17849237

N=C(c1cc(C(N)=O)ccc1F)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 11/20 0.33
PARP1 P09874 2/20 0.33
MAPK14 Q16539 1/20 0.33
GUSB P08236 2/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BCL6 P41182 1/20 0.31
BCOR Q6W2J9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623480 0.89 MAPK14 (0.34) RORCPARP1MAPK14GUSB
SCHEMBL17849205 0.86 DGAT1 (0.32) MAPK14GUSBALDH1A1
SCHEMBL17849236 0.86 RORC (0.36) RORCPARP1MAPK14
SCHEMBL16623600 0.82 TYK2 (0.34) PARP1MAPK14
SCHEMBL16726665 0.81 ALDH2 (0.33)
SCHEMBL16623544 0.80 MEN1 (0.32) MAPK14
SCHEMBL16623547 0.78 SYK (0.36) ALDH1A1
SCHEMBL16623468 0.77 MPO (0.31) RAB9A
SCHEMBL17849215 0.77 CRBN (0.38)
SCHEMBL16726696 0.75 HDAC6 (0.41) RORCALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed