SCHEMBL17849248

SCHEMBL17849248

N=C(c1ccc(N2CCN(C(=O)CO)CC2)cc1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.41
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
AKR1C3 P42330 1/20 0.38
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849249 0.85 EGFR (0.40) EGFRJAK2JAK1ALDH1A1
SCHEMBL17849188 0.85 EGFR (0.40) EGFRJAK2JAK1ALDH1A1
SCHEMBL16623568 0.83 EGFR (0.38) EGFRJAK2JAK1
SCHEMBL16623503 0.80 EGFR (0.35) EGFRJAK2JAK1
SCHEMBL17849221 0.79 EIF2AK2 (0.34) EGFRJAK2JAK1
SCHEMBL16623565 0.78 ALDH1A1 (0.41) ALDH1A1
SCHEMBL16623511 0.77 TYK2 (0.38) JAK2
SCHEMBL17849244 0.77 TYK2 (0.40) EGFRJAK2JAK1ALDH1A1
SCHEMBL18052623 0.77 EGFR (0.36) EGFRJAK2JAK1
SCHEMBL17849247 0.77 MAPT (0.41) EGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed