SCHEMBL17864618

SCHEMBL17864618

Cc1ccc(Cl)c2oc(/C(N)=N/O)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 4/20 0.37
RARB P10826 4/20 0.37
RARG P13631 4/20 0.37
LMNA P02545 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP3A4 P08684 3/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
SLC9A1 P19634 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17843543 0.87 LMNA (0.37) RARARARBRARGLMNAGFER
SCHEMBL19599548 0.87 LMNA (0.37) RARARARBRARGLMNAGFER
SCHEMBL17864569 0.87 LMNA (0.37) RARARARBRARGLMNAGFER
SCHEMBL17843572 0.76 RARA (0.50) RARARARBRARGKMT2AKDM4E
SCHEMBL17864639 0.69 KDM4E (0.38) RARARARBRARGKDM4E
SCHEMBL252154 0.67 ALDH1A1 (0.41) RARARARBRARGGFERKMT2A
SCHEMBL17730412 0.65 LMNA (0.51) LMNAGFERKMT2AL3MBTL1CYP3A4
SCHEMBL4509810 0.65 LMNA (0.51) LMNAGFERKMT2AL3MBTL1CYP3A4
SCHEMBL17737809 0.65 LMNA (0.51) LMNAGFERKMT2AL3MBTL1CYP3A4
SCHEMBL29875584 0.65 TSHR (0.53) LMNAGFERKMT2AL3MBTL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016097004-A1 BICYCLOHETEROARYL-HETEROARYL-BENZOIC ACID COMPOUNDS AS RETINOIC ACID RECEPTOR BETA (RARβ) AGONISTS KING'S COLLEGE LONDON (GB) 2016-06-23 WO disclosed